Hubei, China
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2000000 RMB
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<100 square meters
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North America, Eastern Europe, Southeast Asia, Africa, Mid East, Eastern Asia, Western ...
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Peak season lead time: 3-6 months
Off season lead time: within 15 workdays
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Tianeptine, Tianeptine Sodium, CAS 30123-17-2 manufacturer / supplier in China, offering Best Quality Nootropics Tianeptine Sodium CAS 30123-17-2, Cosmetic Peptide High Quality Myristoyl Tetrapeptide-12 with Best Price 959610-24-3, Pharmaceutical Raw Material Sports Nutritions Powder Ostarine Mk 2866 and so on.

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Best Quality Nootropics Tianeptine Sodium CAS 30123-17-2

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Min. Order: 100 g
Port: Shanghai, China
Production Capacity: 5000kg/M
Payment Terms: T/T, Western Union, Paypal, Money Gram
Powder: Yes
Customized: Non-Customized
Certification: GMP, HSE, ISO 9001, USP, BP
Suitable for: Elderly, Children, Adult
State: Solid
Purity: >99%

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Basic Info

Model NO.
Tianeptine Sodium
Function
Antidepressant
Appearance
White Powder
Molecular Weight
458.93
Trademark
W&Z
Transport Package
FedEx, TNT, EMS, DHL
Specification
Medicine Grade
Origin
Hubei Wu Han
Product Description
Best Quality Nootropics Tianeptine Sodium CAS 30123-17-2


Tianeptine sodium salt  CAS  30123-17-2
Tianeptine sulfate CAS : 1224690-84-9
Tianeptine (Tianeptine Free Acid ) CAS : 66981-73-5



Quick Details for TIANEPTINE SODIUM

Product Name: Tianeptine sodium salt 
Synonyms: TIANEPTINE SODIUM;TIANEPTINE SODIUM SALT;sodium 7-((3-chloro-6,11-dihydro-6-methyldibenzo(c,f)(1,2)thiazepin-11-yl)amino)heptanoate s,s-dioxide;7-[(3-Chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic Acid S,S-Dioxide Sodium Salt;S-1574;Stablon;7-[(3-chloro-6,11-dihydro-6-methyl-dibenzo[c,f][1,2]thiazepine-11-yl)amino]heptanoic acid s,s dioxide sodium salt;Sodium 7-((3-chloro-6,11-dihydro-6-methyldibenzo(c,f)(1,2)thiazepin-11-yl)amino)heptanoate S,S-dioxide 
CAS: 30123-17-2 
MF: C21H24ClN2NaO4S 
MW: 458.93 
EINECS: 250-059-3 
Product Categories: Intermediates & Fine Chemicals;Pharmaceuticals;Heterocycles;Sulfur & Selenium Compounds;Stablon, Coaxil, Tatinol;API;Inhibitors 
Melting point : 1800C 
Storage temp. : Desiccate at RT
Chemical Properties : White to Yellowish Powder 
Usage : Tricyclic compound with psychostimulant, anti-ulcer and anti-emetic properties. Antidepressant 
Usage : Tianeptine (INN) (Stablon, Coaxil, Tatinol) is a selective serotonin reuptake enhancer (SSRE) drug used for treating major depressive episodes (mild, moderate, or severe).  


Tianeptine sodium Description

Tianeptine (brand names Stablon, Coaxil, Tatinol, Tianeurax and Salymbra) is a drug used primarily in the treatment of major depressive disorder, although it may also be used to treat asthma or irritable bowel syndrome. Chemically it is a tricyclic antidepressant (TCA), but it has different pharmacological properties than typical TCAs as recent research suggests that tianeptine produces its antidepressant effects through indirect alteration of glutamate receptor activity (i.e., AMPA receptors and NMDA receptors) and release of BDNF, in turn affecting neural plasticity.

Tianeptine has antidepressant and anxiolytic (anti-anxiety) properties with a relative lack of sedative, anticholinergic and cardiovascular adverse effects,[citation needed] thus suggesting it is particularly suitable for use in the elderly and in those following alcohol withdrawal; such persons can be more sensitive to the adverse effects of psychotropic drugs. Recent results indicate possible anticonvulsant (anti-seizure) and analgesic (painkilling) activity of tianeptine via immediate or downstream modulation of adenosine A1 receptors (as the effects could be experimentally blocked by antagonists of this receptor).


Medical uses of Tianeptine sodium

Tianeptine shows efficacy against serious depressive episodes (major depression), comparable to amitriptyline, imipramine and fluoxetine, but with significantly fewer side effects. It was shown to be more effective than maprotiline in a group of people with co-existing depression and anxiety. Tianeptine also displays significant anxiolytic properties and is useful in treating a spectrum of anxiety disorders including panic disorder, as evidenced by a study in which those administered 35% CO2 gas (carbogen) on paroxetine or tianeptine therapy showed equivalent panic-blocking effects. Like many antidepressants (including bupropion, the selective serotonin reuptake inhibitors, the serotonin-norepinephrine reuptake inhibitors, moclobemide and numerous others) it may also have a beneficial effect on cognition in people with depression-induced cognitive dysfunction.


Tianeptine sodium Side effects

Compared to other TCAs it produces significantly fewer cardiovascular, anticholinergic (like dry mouth or constipation), sedative and appetite-stimulating effects. A recent review found that it was amongst the antidepressants most prone to causing hepatotoxicity (liver damage), although the evidence to support this concern was of limited quality. Although not well studied with tianeptine, it has been shown for tricyclic antidepressants that they may cause cardiac arrhythmias.


 COA
 
Product NameTianeptine sodium
Batch No.160625Mfg. date2016-6-25
Test Date2016-6-25Exp. date2018-6-24
TestsSpecificationsResults
DescriptionWhite to yellowish powder, very hygroscopic.Off-white powder, very hygroscopic.
SolubilityFreetly soluble In water and methanol and dichloromethaneComplies
Identification(1)By IR, To match with working standardComplies
(2)It gives reaction of sodiumComplies
Impurities A≤0.1%Not detected
Related compoundsAny impurity ≤0.1%<0.1%
Total impurities ≤0.4%0.25%
Residual SolventsAcetidin≤ 0.5%Not detected
Dichloromethane≤ 0.06%Not detected
Methanol≤ 0.3%Not detected
Acetone ≤ 0.5%Not detected
Acetonitrile≤0.041%Not detected
Ethanol≤0.5%0.04%
N, N-dimethylformamide≤0.088%Not detected
Water≤ 5.0%1.38%
Assay99.0%-101.0%(On anhydrous basis)99.98%
ConclusionConform to EP8.0
 
Related Products Specifications


Tianeptine sodium salt  CAS  30123-17-2
Tianeptine sulfate CAS : 1224690-84-9
Tianeptine (Tianeptine Free Acid ) CAS : 66981-73-5
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